acrR

Overview

Drug Classes
Fluoroquinolone, Tigecycline, norfloxacin|ciprofloxacin, Norfloxacin, Ciprofloxacin
Organisms
Klebsiella pneumoniae, Escherichia coli
Papers
4
Mutations
29
Mutations29
Nucleotide ChangeProtein ChangeTypeEffect on FunctionResistance ToYearPaperStatus
-F197I--
Fluoroquinolone
2003

Role of AcrR and ramA in fluoroquinolone resistance in clinical Klebsiella pneumoniae isolates from Singapore.

PMID: 12936981
Not Validated
-A20T--
Fluoroquinolone
2003

Role of AcrR and ramA in fluoroquinolone resistance in clinical Klebsiella pneumoniae isolates from Singapore.

PMID: 12936981
Not Validated
-G121*--
Tigecycline
2017

Tigecycline Susceptibility and Molecular Resistance Mechanisms Among Clinical Klebsiella pneumoniae Strains Isolated During Non-Tigecycline Treatment.

PMID: 27219271
Not Validated
-E122K--
Tigecycline
2017

Tigecycline Susceptibility and Molecular Resistance Mechanisms Among Clinical Klebsiella pneumoniae Strains Isolated During Non-Tigecycline Treatment.

PMID: 27219271
Not Validated
-L195V--
Fluoroquinolone
2003

Role of AcrR and ramA in fluoroquinolone resistance in clinical Klebsiella pneumoniae isolates from Singapore.

PMID: 12936981
Not Validated
-M123*--
Tigecycline
2017

Tigecycline Susceptibility and Molecular Resistance Mechanisms Among Clinical Klebsiella pneumoniae Strains Isolated During Non-Tigecycline Treatment.

PMID: 27219271
Not Validated
-L197L--
Fluoroquinolone
2003

Role of AcrR and ramA in fluoroquinolone resistance in clinical Klebsiella pneumoniae isolates from Singapore.

PMID: 12936981
Not Validated
-P161R--
Fluoroquinolone
2003

Role of AcrR and ramA in fluoroquinolone resistance in clinical Klebsiella pneumoniae isolates from Singapore.

PMID: 12936981
Not Validated
-G164A--
Fluoroquinolone
2003

Role of AcrR and ramA in fluoroquinolone resistance in clinical Klebsiella pneumoniae isolates from Singapore.

PMID: 12936981
Not Validated
-F204L--
Tigecycline
2017

Roles of ramR and tet(A) Mutations in Conferring Tigecycline Resistance in Carbapenem-Resistant Klebsiella pneumoniae Clinical Isolates.

PMID: 28533243
Not Validated
-R173G--
Fluoroquinolone
2003

Role of AcrR and ramA in fluoroquinolone resistance in clinical Klebsiella pneumoniae isolates from Singapore.

PMID: 12936981
Not Validated
-A151V--
Fluoroquinolone
2003

Role of AcrR and ramA in fluoroquinolone resistance in clinical Klebsiella pneumoniae isolates from Singapore.

PMID: 12936981
Not Validated
-K201M--
Fluoroquinolone
2003

Role of AcrR and ramA in fluoroquinolone resistance in clinical Klebsiella pneumoniae isolates from Singapore.

PMID: 12936981
Not Validated
-G121V--
Tigecycline
2017

Tigecycline Susceptibility and Molecular Resistance Mechanisms Among Clinical Klebsiella pneumoniae Strains Isolated During Non-Tigecycline Treatment.

PMID: 27219271
Not Validated
-F172S--
Fluoroquinolone
2003

Role of AcrR and ramA in fluoroquinolone resistance in clinical Klebsiella pneumoniae isolates from Singapore.

PMID: 12936981
Not Validated
A147CK146T--
norfloxacin|ciprofloxacin
2003

Mutation rate and evolution of fluoroquinolone resistance in Escherichia coli isolates from patients with urinary tract infections.

PMID: 14506034
Not Validated
A16TI16F--
norfloxacin|ciprofloxacin
2003

Mutation rate and evolution of fluoroquinolone resistance in Escherichia coli isolates from patients with urinary tract infections.

PMID: 14506034
Not Validated
A62TI62F--
norfloxacin|ciprofloxacin
2003

Mutation rate and evolution of fluoroquinolone resistance in Escherichia coli isolates from patients with urinary tract infections.

PMID: 14506034
Not Validated
A63GK62R--
norfloxacin|ciprofloxacin
2003

Mutation rate and evolution of fluoroquinolone resistance in Escherichia coli isolates from patients with urinary tract infections.

PMID: 14506034
Not Validated
C156TP155L--
norfloxacin|ciprofloxacin
2003

Mutation rate and evolution of fluoroquinolone resistance in Escherichia coli isolates from patients with urinary tract infections.

PMID: 14506034
Not Validated
C6AT5N--
norfloxacin|ciprofloxacin
2003

Mutation rate and evolution of fluoroquinolone resistance in Escherichia coli isolates from patients with urinary tract infections.

PMID: 14506034
Not Validated
del382CAGGCCCAGCGGCAG---
Norfloxacin, Ciprofloxacin
2003

Role of AcrR and ramA in fluoroquinolone resistance in clinical Klebsiella pneumoniae isolates from Singapore.

PMID: 12936981
Not Validated
del430ACCTTGAAAGAG---
Norfloxacin, Ciprofloxacin
2003

Role of AcrR and ramA in fluoroquinolone resistance in clinical Klebsiella pneumoniae isolates from Singapore.

PMID: 12936981
Not Validated
G125AV125I--
norfloxacin|ciprofloxacin
2003

Mutation rate and evolution of fluoroquinolone resistance in Escherichia coli isolates from patients with urinary tract infections.

PMID: 14506034
Not Validated
G79AV79I--
norfloxacin|ciprofloxacin
2003

Mutation rate and evolution of fluoroquinolone resistance in Escherichia coli isolates from patients with urinary tract infections.

PMID: 14506034
Not Validated
T202GM201R--
norfloxacin|ciprofloxacin
2003

Mutation rate and evolution of fluoroquinolone resistance in Escherichia coli isolates from patients with urinary tract infections.

PMID: 14506034
Not Validated
T24CF24L--
norfloxacin|ciprofloxacin
2003

Mutation rate and evolution of fluoroquinolone resistance in Escherichia coli isolates from patients with urinary tract infections.

PMID: 14506034
Not Validated
T25CS25P--
norfloxacin|ciprofloxacin
2003

Mutation rate and evolution of fluoroquinolone resistance in Escherichia coli isolates from patients with urinary tract infections.

PMID: 14506034
Not Validated
T47GC47G--
norfloxacin|ciprofloxacin
2003

Mutation rate and evolution of fluoroquinolone resistance in Escherichia coli isolates from patients with urinary tract infections.

PMID: 14506034
Not Validated
Papers4
1

Role of AcrR and ramA in fluoroquinolone resistance in clinical Klebsiella pneumoniae isolates from Singapore.

PMID 12936981 · 2003

Under development. Phenotype should be used with caution.

Mutation Information

Gene Name
acrR
Protein Change
F197I

Confers Resistance To

Fluoroquinolone

Organisms Observed In

Klebsiella pneumoniae
2

Role of AcrR and ramA in fluoroquinolone resistance in clinical Klebsiella pneumoniae isolates from Singapore.

PMID 12936981 · 2003

Under development. Phenotype should be used with caution.

Mutation Information

Gene Name
acrR
Protein Change
A20T

Confers Resistance To

Fluoroquinolone

Organisms Observed In

Klebsiella pneumoniae
3

Tigecycline Susceptibility and Molecular Resistance Mechanisms Among Clinical Klebsiella pneumoniae Strains Isolated During Non-Tigecycline Treatment.

PMID 27219271 · 2017

Under development. Phenotype should be used with caution.

Mutation Information

Gene Name
acrR
Protein Change
G121*

Confers Resistance To

Tigecycline

Organisms Observed In

Klebsiella pneumoniae
4

Tigecycline Susceptibility and Molecular Resistance Mechanisms Among Clinical Klebsiella pneumoniae Strains Isolated During Non-Tigecycline Treatment.

PMID 27219271 · 2017

Under development. Phenotype should be used with caution.

Mutation Information

Gene Name
acrR
Protein Change
E122K

Confers Resistance To

Tigecycline

Organisms Observed In

Klebsiella pneumoniae
5

Role of AcrR and ramA in fluoroquinolone resistance in clinical Klebsiella pneumoniae isolates from Singapore.

PMID 12936981 · 2003

Under development. Phenotype should be used with caution.

Mutation Information

Gene Name
acrR
Protein Change
L195V

Confers Resistance To

Fluoroquinolone

Organisms Observed In

Klebsiella pneumoniae
6

Tigecycline Susceptibility and Molecular Resistance Mechanisms Among Clinical Klebsiella pneumoniae Strains Isolated During Non-Tigecycline Treatment.

PMID 27219271 · 2017

Under development. Phenotype should be used with caution.

Mutation Information

Gene Name
acrR
Protein Change
M123*

Confers Resistance To

Tigecycline

Organisms Observed In

Klebsiella pneumoniae
7

Role of AcrR and ramA in fluoroquinolone resistance in clinical Klebsiella pneumoniae isolates from Singapore.

PMID 12936981 · 2003

Under development. Phenotype should be used with caution.

Mutation Information

Gene Name
acrR
Protein Change
L197L

Confers Resistance To

Fluoroquinolone

Organisms Observed In

Klebsiella pneumoniae
8

Role of AcrR and ramA in fluoroquinolone resistance in clinical Klebsiella pneumoniae isolates from Singapore.

PMID 12936981 · 2003

Under development. Phenotype should be used with caution.

Mutation Information

Gene Name
acrR
Protein Change
P161R

Confers Resistance To

Fluoroquinolone

Organisms Observed In

Klebsiella pneumoniae
9

Role of AcrR and ramA in fluoroquinolone resistance in clinical Klebsiella pneumoniae isolates from Singapore.

PMID 12936981 · 2003

Under development. Phenotype should be used with caution.

Mutation Information

Gene Name
acrR
Protein Change
G164A

Confers Resistance To

Fluoroquinolone

Organisms Observed In

Klebsiella pneumoniae
10

Roles of ramR and tet(A) Mutations in Conferring Tigecycline Resistance in Carbapenem-Resistant Klebsiella pneumoniae Clinical Isolates.

PMID 28533243 · 2017

Under development. Phenotype should be used with caution.

Mutation Information

Gene Name
acrR
Protein Change
F204L

Confers Resistance To

Tigecycline

Organisms Observed In

Klebsiella pneumoniae
11

Role of AcrR and ramA in fluoroquinolone resistance in clinical Klebsiella pneumoniae isolates from Singapore.

PMID 12936981 · 2003

Under development. Phenotype should be used with caution.

Mutation Information

Gene Name
acrR
Protein Change
R173G

Confers Resistance To

Fluoroquinolone

Organisms Observed In

Klebsiella pneumoniae
12

Role of AcrR and ramA in fluoroquinolone resistance in clinical Klebsiella pneumoniae isolates from Singapore.

PMID 12936981 · 2003

Under development. Phenotype should be used with caution.

Mutation Information

Gene Name
acrR
Protein Change
A151V

Confers Resistance To

Fluoroquinolone

Organisms Observed In

Klebsiella pneumoniae
13

Role of AcrR and ramA in fluoroquinolone resistance in clinical Klebsiella pneumoniae isolates from Singapore.

PMID 12936981 · 2003

Under development. Phenotype should be used with caution.

Mutation Information

Gene Name
acrR
Protein Change
K201M

Confers Resistance To

Fluoroquinolone

Organisms Observed In

Klebsiella pneumoniae
14

Tigecycline Susceptibility and Molecular Resistance Mechanisms Among Clinical Klebsiella pneumoniae Strains Isolated During Non-Tigecycline Treatment.

PMID 27219271 · 2017

Under development. Phenotype should be used with caution.

Mutation Information

Gene Name
acrR
Protein Change
G121V

Confers Resistance To

Tigecycline

Organisms Observed In

Klebsiella pneumoniae
15

Role of AcrR and ramA in fluoroquinolone resistance in clinical Klebsiella pneumoniae isolates from Singapore.

PMID 12936981 · 2003

Under development. Phenotype should be used with caution.

Mutation Information

Gene Name
acrR
Protein Change
F172S

Confers Resistance To

Fluoroquinolone

Organisms Observed In

Klebsiella pneumoniae
16

Mutation rate and evolution of fluoroquinolone resistance in Escherichia coli isolates from patients with urinary tract infections.

PMID 14506034 · 2003

Mutation Information

Gene Name
acrR
Nucleotide Change
A147C
Protein Change
K146T

Confers Resistance To

norfloxacin|ciprofloxacin

Organisms Observed In

Escherichia coli
17

Mutation rate and evolution of fluoroquinolone resistance in Escherichia coli isolates from patients with urinary tract infections.

PMID 14506034 · 2003

Mutation Information

Gene Name
acrR
Nucleotide Change
A16T
Protein Change
I16F

Confers Resistance To

norfloxacin|ciprofloxacin

Organisms Observed In

Escherichia coli
18

Mutation rate and evolution of fluoroquinolone resistance in Escherichia coli isolates from patients with urinary tract infections.

PMID 14506034 · 2003

Mutation Information

Gene Name
acrR
Nucleotide Change
A62T
Protein Change
I62F

Confers Resistance To

norfloxacin|ciprofloxacin

Organisms Observed In

Escherichia coli
19

Mutation rate and evolution of fluoroquinolone resistance in Escherichia coli isolates from patients with urinary tract infections.

PMID 14506034 · 2003

Mutation Information

Gene Name
acrR
Nucleotide Change
A63G
Protein Change
K62R

Confers Resistance To

norfloxacin|ciprofloxacin

Organisms Observed In

Escherichia coli
20

Mutation rate and evolution of fluoroquinolone resistance in Escherichia coli isolates from patients with urinary tract infections.

PMID 14506034 · 2003

Mutation Information

Gene Name
acrR
Nucleotide Change
C156T
Protein Change
P155L

Confers Resistance To

norfloxacin|ciprofloxacin

Organisms Observed In

Escherichia coli
21

Mutation rate and evolution of fluoroquinolone resistance in Escherichia coli isolates from patients with urinary tract infections.

PMID 14506034 · 2003

Mutation Information

Gene Name
acrR
Nucleotide Change
C6A
Protein Change
T5N

Confers Resistance To

norfloxacin|ciprofloxacin

Organisms Observed In

Escherichia coli
22

Role of AcrR and ramA in fluoroquinolone resistance in clinical Klebsiella pneumoniae isolates from Singapore.

PMID 12936981 · 2003

Under development. Phenotype should be used with caution.

Mutation Information

Gene Name
acrR
Nucleotide Change
del382CAGGCCCAGCGGCAG

Confers Resistance To

Norfloxacin, Ciprofloxacin

Organisms Observed In

Klebsiella pneumoniae
23

Role of AcrR and ramA in fluoroquinolone resistance in clinical Klebsiella pneumoniae isolates from Singapore.

PMID 12936981 · 2003

Under development. Phenotype should be used with caution.

Mutation Information

Gene Name
acrR
Nucleotide Change
del430ACCTTGAAAGAG

Confers Resistance To

Norfloxacin, Ciprofloxacin

Organisms Observed In

Klebsiella pneumoniae
24

Mutation rate and evolution of fluoroquinolone resistance in Escherichia coli isolates from patients with urinary tract infections.

PMID 14506034 · 2003

Mutation Information

Gene Name
acrR
Nucleotide Change
G125A
Protein Change
V125I

Confers Resistance To

norfloxacin|ciprofloxacin

Organisms Observed In

Escherichia coli
25

Mutation rate and evolution of fluoroquinolone resistance in Escherichia coli isolates from patients with urinary tract infections.

PMID 14506034 · 2003

Mutation Information

Gene Name
acrR
Nucleotide Change
G79A
Protein Change
V79I

Confers Resistance To

norfloxacin|ciprofloxacin

Organisms Observed In

Escherichia coli
26

Mutation rate and evolution of fluoroquinolone resistance in Escherichia coli isolates from patients with urinary tract infections.

PMID 14506034 · 2003

Mutation Information

Gene Name
acrR
Nucleotide Change
T202G
Protein Change
M201R

Confers Resistance To

norfloxacin|ciprofloxacin

Organisms Observed In

Escherichia coli
27

Mutation rate and evolution of fluoroquinolone resistance in Escherichia coli isolates from patients with urinary tract infections.

PMID 14506034 · 2003

Mutation Information

Gene Name
acrR
Nucleotide Change
T24C
Protein Change
F24L

Confers Resistance To

norfloxacin|ciprofloxacin

Organisms Observed In

Escherichia coli
28

Mutation rate and evolution of fluoroquinolone resistance in Escherichia coli isolates from patients with urinary tract infections.

PMID 14506034 · 2003

Mutation Information

Gene Name
acrR
Nucleotide Change
T25C
Protein Change
S25P

Confers Resistance To

norfloxacin|ciprofloxacin

Organisms Observed In

Escherichia coli
29

Mutation rate and evolution of fluoroquinolone resistance in Escherichia coli isolates from patients with urinary tract infections.

PMID 14506034 · 2003

Mutation Information

Gene Name
acrR
Nucleotide Change
T47G
Protein Change
C47G

Confers Resistance To

norfloxacin|ciprofloxacin

Organisms Observed In

Escherichia coli